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Mefloquine diacetate

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Identification
Molecular formula
C27H32N4O4
CAS number
38077-85-5
IUPAC name
1-[10-(4-amino-2-methyl-quinolin-1-ium-1-yl)decyl]-2-methyl-quinolin-1-ium-4-amine;diacetate
State
State

This compound is typically found in its solid form at room temperature, often as a powder. Its solid state is a common characteristic due to its crystalline nature.

Melting point (Celsius)
106.00
Melting point (Kelvin)
379.15
Boiling point (Celsius)
196.00
Boiling point (Kelvin)
469.15
General information
Molecular weight
622.71g/mol
Molar mass
622.7050g/mol
Density
1.2800g/cm3
Appearence

Mefloquine diacetate generally appears as an off-white to slightly yellow crystalline powder. It is recognized for its characteristic crystalline form which may vary slightly in shade depending on purity and batch conditions.

Comment on solubility

Solubility of 1-[10-(4-amino-2-methyl-quinolin-1-ium-1-yl)decyl]-2-methyl-quinolin-1-ium-4-amine; diacetate

The solubility of 1-[10-(4-amino-2-methyl-quinolin-1-ium-1-yl)decyl]-2-methyl-quinolin-1-ium-4-amine; diacetate can be influenced by several factors which reflect its complex structure, particularly the presence of quinoline moieties and ionic interactions from the diacetate component. Here are some key points to consider:

  • Polarity: The quinoline rings contribute to the overall polarity of the molecule. Molecules with higher polarity tend to have better solubility in polar solvents, such as water.
  • Ionic Nature: The diacetate part of the compound may enhance its solubility in aqueous solutions due to ionic interactions, making it more soluble compared to neutral compounds.
  • Solvent Selection: The solubility can vary significantly between different solvents. For example:
    • In polar solvents (e.g., water, ethanol) - Enhanced solubility.
    • In non-polar solvents (e.g., hexane) - Reduced solubility.
  • Temperature Effect: Like many chemical compounds, the solubility may increase with temperature, allowing for greater molecular motion and interaction with solvents.

In summary, while the solubility of this quinolinium compound is likely favorable in polar environments due to its ionic and polar nature, precise quantitative solubility values would require experimental determination. Understanding the “like dissolves like” principle is crucial for predicting its behavior in various solvent systems.

Interesting facts

Interesting Facts about 1-[10-(4-amino-2-methyl-quinolin-1-ium-1-yl)decyl]-2-methyl-quinolin-1-ium-4-amine; diacetate

This fascinating compound, known for its complex structure, is a derivative of quinoline, a heterocyclic aromatic organic compound that has piqued the interest of scientists across various fields. Here are some noteworthy facts about this intriguing compound:

  • Quinoline Derivative: The structure incorporates quinoline moieties, which are known for their biological significance, particularly in medicinal chemistry where they exhibit antimicrobial and antimalarial properties.
  • Distinctive Amino Groups: The presence of amino groups enhances the compound's potential as a versatile building block for synthesizing more complex molecules.
  • Decyl Chain Influence: The long decyl chain in the compound increases its lipophilicity, which can significantly influence its interactions with biological membranes, thus impacting its efficacy in medicinal applications.
  • Potential Applications: Given its unique structure, this compound could be explored for use in:
    • Drug development, especially targeted therapies
    • Fluorescent probes for biological imaging
    • Environmental chemistry for dye-sensitized solar cells
  • Research Interest: As scientists continue to investigate the properties of compounds similar to this, it presents exciting opportunities for new discoveries in pharmacology and material sciences.

Overall, 1-[10-(4-amino-2-methyl-quinolin-1-ium-1-yl)decyl]-2-methyl-quinolin-1-ium-4-amine; diacetate is more than just a chemical formula; it's a potential key to unlocking new solutions in various scientific fields, illustrating the intricate relationship between molecular structure and function.

Synonyms
DEQUALINIUM ACETATE
Dequadin acetate
Decalinium acetate
EINECS 223-712-5
UNII-P8W4UX112S
Acetate, Dequalinium
P8W4UX112S
1,1'-Decamethylenebis(4-aminoquinaldinium acetate)
1,1'-(decane-1,10-diyl)bis[4-amino-2-methylquinolinium] diacetate
DTXSID80193267
1,1'-(1,10-Decanediyl)bis(4-amino-2-methylquinolinium) diacetate
1,1'-(Decane-1,10-diyl)bis(4-amino-2-methylquinolinium) diacetate
Quinolinium, 1,1'-(1,10-decanediyl)bis(4-amino-2-methyl-, diacetate
DEQUALINIUM ACETATE [WHO-DD]
Quinaldinium, 1,1'-decamethylenebis(4-amino-, diacetate
Dequalinium Diacetate
Diacetate, Dequalinium
DTXCID90115758
DEQUALINIUM ACETATE [INCI]
Quinolinium, 1,1'-(1,10-decanediyl)bis(4-amino-2-methyl-), Diacetate
Quinolinium, 1,1'-(1,10-decanediyl)bis(4-amino-2-methyl-, diacetate (9CI)
4028-98-2
1,1'-(decane-1,10-diyl)bis(4-amino-2-methylquinolin-1-ium) acetate
1-[10-(4-amino-2-methylquinolin-1-ium-1-yl)decyl]-2-methylquinolin-1-ium-4-amine;diacetate
SCHEMBL677152
NS00083541
Q27286389
1,1'-(Decane-1,10-diyl)bis[4-amino-2-methylquinolinium]diacetate