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Carfentanil

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Identification
Molecular formula
C24H30ClN3O3
CAS number
59708-52-0
IUPAC name
1-[3-(3-chlorobenzo[b][1]benzazepin-11-yl)propyl]-4-(dimethylamino)piperidine-4-carboxamide
State
State

At room temperature, carfentanil is in a solid state, typically found as a crystalline powder.

Melting point (Celsius)
200.00
Melting point (Kelvin)
473.20
Boiling point (Celsius)
583.30
Boiling point (Kelvin)
856.50
General information
Molecular weight
394.97g/mol
Molar mass
394.9240g/mol
Density
1.3105g/cm3
Appearence

Carfentanil, in its pure form, appears as a white to off-white powder. Due to its extremely high potency, it is typically diluted before handling in practical applications.

Comment on solubility

Solubility of 1-[3-(3-chlorobenzob[1]benzazepin-11-yl)propyl]-4-(dimethylamino)piperidine-4-carboxamide

The solubility of the compound 1-[3-(3-chlorobenzob[1]benzazepin-11-yl)propyl]-4-(dimethylamino)piperidine-4-carboxamide can be influenced by various factors, including its molecular structure, the presence of functional groups, and the solvent used. This compound contains both polar and nonpolar regions, contributing to its moderate solubility characteristics. Here are several important points regarding its solubility:

  • Polarity: The presence of the polar dimethylamino group may enhance solubility in polar solvents, whereas the aromatic systems could limit solubility in aqueous environments.
  • Hydrophilicity vs. Hydrophobicity: The balance between hydrophilic (water-attracting) and hydrophobic (water-repelling) regions plays a critical role in determining solubility, which may be moderate in water.
  • Solvent Compatibility: This compound is likely to be more soluble in organic solvents such as DMSO or ethanol, rather than in water, due to the substantial nonpolar character from its phenyl and piperidine groups.
  • Temperature Effects: The solubility may vary with temperature; generally, an increase in temperature enhances solubility for many compounds.

As a general assessment, studying the specific solubility properties in various solvents can provide a better understanding of this compound's behavior in different chemical environments. Consider conducting empirical measurements for more precise solubility data.

Interesting facts

Interesting Facts About 1-[3-(3-chlorobenzo©[1]benzazepin-11-yl)propyl]-4-(dimethylamino)piperidine-4-carboxamide

This compound is part of a class of chemical entities known for their potential pharmacological activities. Let's explore some captivating aspects of this unique structure:

  • Versatile Structure: The compound features a piperidine ring, which is a five-membered nitrogen-containing structure. This ring system is known for its significant role in various biological activities, making it a valuable scaffold in drug design.
  • Chlorobenzo© Group: The presence of the chlorobenzo[b][1]benzazepin moiety contributes to the unique binding properties of this compound, potentially influencing its interaction with various biological targets.
  • Medical Interest: Compounds that exhibit structural similarities to this molecule have been studied for their effects on the central nervous system, including potential treatments for mood disorders. Continuous research aims to explore their therapeutic potential further.
  • Dimethylamino Functionality: The dimethylamino group enhances the compound's lipophilicity, which might improve its ability to cross biological membranes, a critical factor for drug efficacy.
  • Potential in Medicinal Chemistry: Due to its intricate structure, this compound serves as a lead structure in medicinal chemistry. Scientists continually seek to optimize such compounds for improved biological activity and reduced side effects.

As researchers delve into the complexities of molecules like 1-[3-(3-chlorobenzo©[1]benzazepin-11-yl)propyl]-4-(dimethylamino)piperidine-4-carboxamide, they uncover novel mechanisms of action that may lead to groundbreaking treatments in various fields of medicine. The ongoing exploration of this compound exemplifies the exciting intersection of chemistry and pharmacology.