Interesting facts
Interesting Facts about 2-[4-[3-(2-chlorophenothiazin-10-yl)propyl]piperazin-1-yl]ethyl 3,4,5-trimethoxybenzoate;ethanesulfonic acid
This compound is a fascinating example of a complex pharmaceutical agent that merges elements of organic chemistry with medicinal applications. Here are some key points to consider:
- Multifunctional Structure: The compound features a blend of a chlorophenothiazine moiety and a piperazine ring, which contributes to its pharmacological activity. The trifecta of methoxy groups enhances its lipophilicity, facilitating better biological interactions.
- Pharmaceutical Relevance: Compounds like this are often investigated for their potential therapeutic roles, particularly in psychiatric disorders and as antipsychotics. The inclusion of piperazine units is common in many antidepressants and antipsychotic medications, indicating possible analgesic properties.
- Chlorine Significance: The chlorophenothiazine structure often correlates with heightened therapeutic efficacy and varied side effect profiles. The presence of chlorine atoms can significantly influence the behavior of the compound in biological systems.
- Synthesis & Modification: Researchers constantly seek to optimize such compounds through structural modifications to enhance their effectiveness and reduce adverse effects. This compound exemplifies how small chemical changes can influence biological activity.
- Complex Interactions: The ethyl ester and sulfonic acid components suggest this compound may interact with various biological pathways, potentially offering unique mechanisms of action within the central nervous system.
Overall, the study of 2-[4-[3-(2-chlorophenothiazin-10-yl)propyl]piperazin-1-yl]ethyl 3,4,5-trimethoxybenzoate;ethanesulfonic acid underscores the intricate relationship between chemical structure and biological function in pharmacology. As science continues to unravel the complexities of such compounds, the potential for innovative therapeutic solutions remains an exciting frontier in the field!
Synonyms
Methophenazine diethanesulfonate
Metofenazate diesylate
UNII-YM9W99502E
YM9W99502E
DTXSID30168283
BENZOIC ACID, 3,4,5-TRIMETHOXY-, 2-(4-(3-(2-CHLORO-10H-PHENOTHIAZIN-10-YL)PROPYL)-1-PIPERAZINYL)ETHYL ESTER, ETHANESULFONATE (1:2)
DTXCID8090774
1674-48-2
Benzoic acid, 3,4,5-trimethoxy-, 2-(4-(3-(2-chlorophenothiazin-10-yl)propyl)-1-piperazinyl)ethyl ester, diethanesulfonate
Metofenazate diethanesulfonate
EX-A10637
Q27294589
Solubility of 2-[4-[3-(2-chlorophenothiazin-10-yl)propyl]piperazin-1-yl]ethyl 3,4,5-trimethoxybenzoate;ethanesulfonic acid
The solubility of a chemical compound is a crucial factor in its application and effectiveness, particularly in pharmaceuticals. When considering the solubility of 2-[4-[3-(2-chlorophenothiazin-10-yl)propyl]piperazin-1-yl]ethyl 3,4,5-trimethoxybenzoate;ethanesulfonic acid, several aspects come into play:
Studies indicate that the solubility of this compound in water may not be extensive due to its complex structure, yet it might show good solubility in organic solvents or buffered solutions. Understanding its solubility profile is essential for effective formulation and bioavailability considerations.