Skip to main content

Flupentixol

ADVERTISEMENT
Identification
Molecular formula
C23H25F3NOS
CAS number
2709-56-0
IUPAC name
2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol
State
State

At room temperature, Flupentixol exists as a solid. It is usually processed and delivered in the form of tablets or injectable solutions for pharmacological applications.

Melting point (Celsius)
113.00
Melting point (Kelvin)
386.15
Boiling point (Celsius)
275.00
Boiling point (Kelvin)
548.15
General information
Molecular weight
437.53g/mol
Molar mass
437.5340g/mol
Density
1.3500g/cm3
Appearence

Flupentixol is commonly found as a crystalline powder. It may appear as a white or slightly yellowish powder. It is often used in its dihydrochloride form for medical purposes.

Comment on solubility

Solubility of 2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol

The solubility of a chemical compound is influenced by various factors, including its molecular structure, polarity, and the nature of the solvent. In the case of 2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol, we can make some interesting observations:

  • Polarity: This compound features various functional groups, including an ethanol moiety, which typically enhances solubility in polar solvents due to hydrogen bonding.
  • Hydrophobic sections: The presence of the thioxanthenyl and trifluoromethyl groups may contribute to hydrophobic interactions, complicating solubility in polar environments.
  • Microscopic interactions: The molecular interactions at play can lead to varying solubility behaviors. This compound could exhibit differing levels of solubility in aqueous vs. organic solvents.
  • Temperature dependence: Like many compounds, solubility can also change with temperature—either increasing or decreasing, depending on the specific solvent environment.

To sum up, while the presence of the alcohol group suggests potential for solubility in polar solvents, the bulky and hydrophobic nature of the thioxanthenyl structure and trifluoromethyl group might limit its overall solubility in aqueous solutions. Therefore, experimental solubility testing is recommended to ascertain precise solubility characteristics in various solvent systems.

Interesting facts

Interesting Facts About 2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol

This fascinating compound is a member of the thioxanthenes, a class of compounds known for their complex aromatic structures and significant biological activity. Here are some intriguing facts about this particular molecule:

  • Medicinal Applications: Due to its unique structure, this compound is of interest in pharmacology. Compounds resembling thioxanthene have been investigated for their potential as antipsychotic medications.
  • Fluorine's Role: The presence of the trifluoromethyl group (–CF3) enhances the compound's biological properties and lipophilicity, increasing membrane permeability.
  • Structure-Activity Relationships: Researchers often explore how modifications to the thioxanthenic core influence pharmacological effects, paving the way for the development of novel therapeutic agents.
  • Versatile Substituents: The piperazine moiety in this compound is known for its versatility in medicinal chemistry, often serving as a framework for enhancing drug activities through various substitutions.
  • Research Potential: The compound’s complex structure and unique functional groups make it a prime candidate for further investigation in drug design and synthetic chemistry.

In summary, 2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol serves as an exemplary compound for studying structural effects on biological activity, showcasing the intricate relationship between chemistry and medicinal application. As research evolves, this compound may pave the way for innovative treatments in the field of psychiatry.

Synonyms
Flupentixol
FLUPENTHIXOL
2709-56-0
2-[4-[3-[2-(trifluoromethyl)-9-thioxanthenylidene]propyl]-1-piperazinyl]ethanol
Flupentiol
2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol
Prestwick0_000340
Prestwick1_000340
SPBio_002300
CHEMBL4743867
DTXSID3058749
NJMYODHXAKYRHW-UHFFFAOYSA-N
NS00076284
Q27164953
(ez)-2-[4-[3-[2-(trifluoromethyl)thioxanthen-9-ylidene]propyl]piperazin-1-yl]ethanol