Interesting facts
Interesting Facts About 2-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one
The compound known as 2-chloro-5-[2-(dimethylamino)ethyl]-11H-benzob[1,4]benzodiazepin-6-one is a fascinating member of the benzodiazepine family. Known for its structural complexity and varied applications, this compound captures the attention of chemists and pharmacologists alike.
Applications and Uses
This compound has been studied for various potential applications, including:
- Pharmaceutical Interest: As a benzodiazepine derivative, it is primarily investigated for its anxiolytic and sedative properties.
- Chemical Intermediary: It serves as a versatile building block in organic synthesis, facilitating the development of new therapeutic agents.
- Research Tool: With its unique functional groups, it is useful in exploring interactions within biological systems.
Structure and Properties
The structure of this compound features:
- A chlorine atom that influences the compound's reactivity and biological activity.
- A dimethylaminoethyl side chain that enhances its pharmacological profile.
- A benzodiazepine core that is crucial for its mechanism of action on the central nervous system.
Noteworthy Insights
When studying this compound, researchers often note the following:
- The presence of the benzodiazepine ring contributes to GABA receptor modulation, which is essential in the context of anxiety and sleep disorders.
- Its synthetic pathway often involves multi-step reactions, highlighting the creativity and skill required in organic synthesis.
- Advancements in medicinal chemistry may lead to derivatives with improved efficacy and fewer side effects.
Overall, 2-chloro-5-[2-(dimethylamino)ethyl]-11H-benzob[1,4]benzodiazepin-6-one stands as a prime example of how intricate structures can translate into significant medicinal properties, making it a valuable subject for ongoing scientific research.
Synonyms
Clobenzepam
Clobenzepam [INN]
1159-93-9
Clobenzepamum
Clobenzepamum [INN-Latin]
Tarpan
UNII-0O6W0NP518
BRN 0895864
0O6W0NP518
CLOBENZEPAM [MI]
WA 172
DTXSID50151218
5-24-04-00114 (Beilstein Handbook Reference)
10,11-Dihydro-11-oxo-5H-dibenzo(b,e)(1,4)diazepine, 7-chloro-10-(2'-(dimethylamino)ethyl)-
7-Chlor-10-beta-dimethylamino-aethyl-10,11-dihydro-11-oxo-5H-dibenzo(b,e)(1,4)diazepin
7-Chloro-10-(2-(dimethylamino)ethyl)-5,10-dihydro-11H-dibenzo(b,e)(1,4)diazepin-11-one
Clobenzepamum (INN-Latin)
5H-Dibenzo(b,e)(1,4)diazepin-11-one, 10,11-dihydro-7-chloro-10-(2-(dimethylamino)ethyl)-
DTXCID9073709
2-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one
SCHEMBL142326
CHEMBL2104007
CHEBI:135352
NS00100933
Q5134760
Solubility of 2-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one
The compound 2-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one exhibits intriguing solubility characteristics influenced by its structure. Its solubility can be affected by various factors, including:
Generally, this compound is expected to have:
Overall, the solubility profile of this compound presents both challenges and opportunities for formulation, especially in pharmaceutical applications. As a reminder, solubility is critical for understanding the behavior of compounds in biological systems and their eventual therapeutic efficacy.