Interesting Facts about 9-Chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one
This compound is a member of the benzodiazepine family, which is known for its diverse effects on the central nervous system. Benzodiazepines are primarily recognized for their sedative, anxiolytic, and muscle-relaxant properties.
Chemical Characteristics
- Structure: The unique structure of this compound includes a 9-chloro substitution, which can influence its pharmacological properties compared to other benzodiazepines.
- Side Chain: The presence of the dimethylamino ethyl side chain contributes to its potential potency and binding affinity for GABAA receptors.
- Receptor Interaction: It is suggested that compounds with similar structures can act as agonists at the benzodiazepine site, enhancing the inhibitory effects of gamma-aminobutyric acid (GABA).
Applications
Due to its structural and chemical properties, this compound has potential implications in various fields:
- Pharmaceutical Research: Investigations into its effects may lead to the development of new therapeutic agents for treating anxiety disorders and insomnia.
- Psychoactive Studies: Research into its effects on mood and cognition could provide insights into treatment options for mood disorders.
- Neuroscience: As a model compound, it may be used to study mechanisms of action of various CNS-active molecules.
Fun Fact
This compound illustrates the diversity found within the benzodiazepine class, showcasing the intricate balance between structure and function in medicinal chemistry. As noted by chemists, "The right side group can make all the difference in pharmacological activity and efficacy."
In summary, 9-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one is more than just a chemical entity; it embodies the ongoing quest in the field of pharmacology to understand and manipulate interactions within the nervous system for better therapeutic outcomes.
Solubility of 9-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one
The solubility of 9-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one in various solvents is a critical aspect to consider for its applications and behavior in different environments. Here are some important points regarding its solubility:
In conclusion, the solubility of 9-chloro-5-[2-(dimethylamino)ethyl]-11H-benzo[b][1,4]benzodiazepin-6-one is multifaceted, influenced by solvent choice, temperature, and environmental pH. Understanding these characteristics is vital for its practical uses in pharmaceuticals and related fields.