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Eprosartan

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Identification
Molecular formula
C23H24N2O9
CAS number
133040-01-4
IUPAC name
methyl 2-[[2-[2-[5-[1-(2-aminopropanoylamino)ethyl]-3-benzyl-2,3,6,7-tetrahydroazepin-1-yl]propanoylamino]-3-methyl-butanoyl]amino]-3-methyl-butanoate
State
State

At room temperature, Eprosartan exists as a solid. It is stable and generally found in pharmaceutical preparations as a white to off-white powder. The solid form is chosen for its chemical stability and ease of formulation into dosage forms.

Melting point (Celsius)
248.00
Melting point (Kelvin)
521.15
Boiling point (Celsius)
450.00
Boiling point (Kelvin)
723.15
General information
Molecular weight
424.25g/mol
Molar mass
424.5260g/mol
Density
1.3000g/cm3
Appearence

The compound appears as a white to off-white crystalline powder. It is typically odorless and stable under standard laboratory conditions. The structure is complex due to its benzyl and tetrahydroazepin groups, contributing to its crystalline nature.

Comment on solubility

Solubility of Methyl 2-[[2-[2-[5-[1-(2-aminopropanoylamino)ethyl]-3-benzyl-2,3,6,7-tetrahydroazepin-1-yl]propanoylamino]-3-methyl-butanoyl]amino]-3-methyl-butanoate

The solubility of the compound methyl 2-[[2-[2-[5-[1-(2-aminopropanoylamino)ethyl]-3-benzyl-2,3,6,7-tetrahydroazepin-1-yl]propanoylamino]-3-methyl-butanoyl]amino]-3-methyl-butanoate (C23H24N2O9) can be examined through several important factors:

  • Polarity: With a complex structure and various functional groups, the polarity of this compound is likely to influence its solubility in different solvents.
  • Hydrogen Bonding: The presence of amino groups suggests that hydrogen bonding could enhance solubility in polar solvents, such as water.
  • Solvent Choice: The compound may exhibit differential solubility in organic solvents. For example, it may be more soluble in ethanol or dimethyl sulfoxide (DMSO) compared to non-polar solvents.
  • pH Sensitivity: The amino groups hint at potential pH sensitivity, meaning that solubility could change under acidic or basic conditions.
  • Temperature Influence: Like most compounds, an increase in temperature typically enhances solubility; thus, heating could be beneficial.

In summary, the solubility of this intricate compound is contingent upon its structural features, the nature of the solvent used, and the surrounding environmental conditions. Therefore, it is crucial to consider all these factors when exploring its applications in various biochemical contexts.

Interesting facts

Interesting Facts About Methyl 2-[[2-[2-[5-[1-(2-aminopropanoylamino)ethyl]-3-benzyl-2,3,6,7-tetrahydroazepin-1-yl]propanoylamino]-3-methyl-butanoyl]amino]-3-methyl-butanoate

This complex compound is a fascinating example of how intricate structures in organic chemistry can lead to significant biological properties. Here are some engaging aspects to consider:

  • Structural Complexity: The compound features a highly intricate structure that combines multiple amino acid sequences and a tetrahydroazepine ring. This complexity can lead to unique interactions in biological systems.
  • Applications in Medicinal Chemistry: Compounds related to this structure have been explored for their potential in drug development, particularly as bioactive molecules that may serve as enzyme inhibitors or in targeting specific receptors in the body.
  • Research Significance: Ongoing research is investigating how the specific arrangement of its amino acids influences its activity, stability, and compatibility with various biological targets.
  • Designing Analogues: Chemists are often inspired by such structures to create analogues that might enhance efficacy or reduce side effects in medical therapies.
  • Potential in Neuropeptide Research: The structural moieties in this compound hint at potential roles in neuropeptide pathways, making it a candidate for studying neurobiological processes.

In summary, methyl 2-[[2-[2-[5-[1-(2-aminopropanoylamino)ethyl]-3-benzyl-2,3,6,7-tetrahydroazepin-1-yl]propanoylamino]-3-methyl-butanoyl]amino]-3-methyl-butanoate is not just a compound with a long name; it is a potential key player in the quest for novel therapeutic agents. Its chemical beauty and potential applications make it a compelling subject for ongoing research!