Cefditoren pivoxil

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Identification

Molecular formula
C25H28N6O7S3
CAS Number
117467-28-4
IUPAC Name
2,2-dimethylpropanoyloxymethyl 7-[[2-(2-aminothiazol-4-yl)-2-methoxyimino-acetyl]amino]-3-[(5-methyltetrazol-2-yl)methyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylate
Molecular Weight
668.76g/mol
Melting Point
(Celsius)
Boiling Point
(Celsius)
Density
1.4400g/cm3
Appearance
can be refined more under different conditions where it can appear slightly yellowish.
Synonyms
cefteram pivoxil
Interesting facts

Interesting Facts about 2,2-Dimethylpropanoyloxymethyl 7-[[2-(2-Aminothiazol-4-yl)-2-Methoxyimino-Acetyl]amino]-3-[(5-Methyltetrazol-2-yl)methyl]-8-Oxo-5-Thia-1-Azabicyclo[4.2.0]oct-2-ene-2-Carboxylate

This compound, with its complex structure, showcases the fascinating world of medicinal chemistry. Here are some intriguing aspects:

  • Mechanism of Action: This compound is part of a novel class of antibiotics, which work by inhibiting bacterial cell wall synthesis. Its unique structure allows it to target specific pathogens more effectively.
  • Bioactivity: The incorporation of thiazole and tetrazole rings is significant because these motifs often exhibit enhanced bioactivity, aiding in the overall efficacy of therapeutic agents.
  • Analog Development: Chemists often synthesize analogs of this compound to enhance their pharmacological profiles. *This iterative process is crucial for drug development, leading to improved selectivity and lower side effects.*
  • Structure-Activity Relationship (SAR): Researchers study the relationship between the chemical structure and its biological activity, which serves as a pathway to design even more potent compounds.
  • Synthesis Challenges: The synthesis of this compound entails multiple steps requiring precision and expertise. *Overcoming these challenges represents a significant achievement in organic synthesis.*
  • Potential Applications: Beyond antibiotics, there is potential for this compound or its derivatives to be explored in anti-cancer therapies due to similar mechanisms observed in camptothecin and other anti-cancer drugs.

In summary, this compound is not just a chemical entity; it embodies the fusion of structure, function, and a promising future in biomedical applications. *As scientists continue to unravel its potential, the excitement in the lab is palpable.*

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