Fluoroethyl piperidinyl quinazoline dione

ADVERTISEMENT

Identification

Molecular formula
C21H20FN3O3
CAS Number
198560-81-7
IUPAC Name
3-[2-[4-(4-fluorobenzoyl)-1-piperidyl]ethyl]-1H-quinazoline-2,4-dione
Molecular Weight
368.40g/mol
Melting Point
(Celsius)
Boiling Point
(Celsius)
Density
1.3765g/cm3
Appearance
may vary slightly depending on the degree of purity and the form in which it is synthesized or stored.
Synonyms
Ketanserin
Interesting facts

Interesting Facts about 3-[2-[4-(4-fluorobenzoyl)-1-piperidyl]ethyl]-1H-quinazoline-2,4-dione

This intriguing compound, often referred to in research circles, has garnered attention for its potential applications in medicinal chemistry. Here are some key points that highlight its significance:

  • Pharmaceutical Relevance: Compounds with a quinazoline structure are frequently studied for their biological activity. This specific compound is believed to exhibit promising antitumor properties, making it a topic of interest in cancer research.
  • Fluorine's Role: The presence of the fluorine atom in this compound greatly enhances its lipophilicity and metabolic stability, which are critical factors in drug design.
  • Complex Structure: The incorporation of a piperidine ring and a benzoyl moiety enhances the compound's interactions with biological targets, offering potential pathways for therapeutic action.
  • Research Opportunities: Due to its unique structure, this compound serves as a versatile scaffold for the synthesis of derivatives that may have improved efficacy or reduced side effects.
  • Structure-Activity Relationship (SAR): Investigating the SAR of compounds like this one helps chemists understand which structural elements contribute to biological activity, ultimately guiding the development of more effective drugs.

Overall, the study of this compound is a fine illustration of how intricate molecular designs can lead to significant advancements in medical science. As research progresses, this compound may unlock new possibilities in targeted therapy.

ADVERTISEMENT